THE ORGANIC CHEMISTRY OF DRUG SYNTHESIS -- CONTENTS -- Preface -- 1 OPEN-CHAIN COMPOUNDS -- 1. Peptidomimetic Compounds -- A. Antiviral Protease Inhibitors -- 1. Human Immunodeficiency Virus -- 2. Human Rhinovirus -- 2. Miscellaneous Peptidomimetic Compounds -- References -- 2 ALICYCLIC COMPOUNDS -- 1. Monocyclic Compounds -- A. Prostaglandins -- B. Antiviral Agents -- C. Miscellaneous Monocyclic Compounds -- 2. Polycyclic Compounds: Steroids -- A. 19-Nor Steroids -- B. Corticosteroid Related Compounds -- 3. Polycyclic Compounds -- References -- 3 MONOCYCLIC AROMATIC COMPOUNDS -- 1. Arylcarbonyl Derivatives -- 2. Biphenyls -- 3. Compounds Related to Aniline -- 4. Compounds Related to Arylsulfonic Acids -- 5. Diarylmethanes -- 6. Miscellaneous Monocyclic Aromatic Compounds -- References -- 4 CARBOCYCLIC COMPOUNDS FUSED TO A BENZENE RING -- 1. Indenes -- 2. Naphthalenes -- 3. Tetrahydronaphthalenes -- 4. Other benzofused carbocyclic compounds -- References -- 5 FIVE-MEMBERED HETEROCYCLES -- 1. Compounds with One Heteroatom -- 2. Compounds with Two Heteroatoms -- A. Oxazole and Isoxazoles -- B. Imidazoles and a Pyrrazole -- C. Thiazoles -- D. Triazoles -- E. Tetrazoles -- References -- 6 SIX-MEMBERED HETEROCYCLES -- 1. Compounds with One Heteroatom -- A. Pyridines -- B. Reduced Pyridines -- C. Miscellaneous -- 2. Compounds with Two Heteroatoms -- A. Pyrimidines -- B. Miscellaneous Six-Membered Heterocycles -- References -- 7 FIVE-MEMBERED HETEROCYCLES FUSED TO ONE BENZENE RING -- 1. Compounds with One Heteroatom -- A. Benzofurans -- B. Indoles -- C. Indolones -- D. Miscellaneous Compounds with One Heteroatom -- 2. Five-Membered Rings with Two Heterocyclic Atoms -- A. Benzimidazoles -- B. Miscellaneous Compounds -- References -- 8 SIX-MEMBERED HETEROCYCLES FUSED TO ONE BENZENE RING -- 1. Compounds with One Heteroatom -- A. Benzopyrans.

B. Quinolines and Their Derivatives -- C. Quinolone Antibacterial Agents -- 2. Compounds with Two Heteroatoms -- A. Benzoxazines -- B. Quinazolines -- C. Miscellaneous Benzo-Fused Heterocycles -- References -- 9 BICYCLIC FUSED HETEROCYCLES -- 1. Compounds with Five-Membered Rings Fused to Six-Membered Rings -- A. Compounds with Two Heteroatoms -- B. Compounds with Three Heteroatoms -- C. Compounds with Four Heteroatoms -- 2. Compounds with Two Fused Six-Membered Rings -- 3. Miscellaneous Compounds with Two Fused Heterocyclic Rings: Beta Lactams -- References -- 10 POLYCYCLIC FUSED HETEROCYCLES -- 1. Compounds with Three Fused Rings -- 2. Compounds with Four Fused Rings -- 3. Compounds with Five or More Fused Rings: Camptothecins -- References -- Subject Index -- Cross Index of Biological Activity -- Cumulative Index.